Neurokinin Receptor Inhibitors

NK1

NK2

NK3

Neurokinin Receptor Inhibitors, Agonists, Antagonists & Modulators

Product Name	NK1	NK2	NK3	Purity
Substance P	NK1			99.82%
Fezolinetant			NK3	99.19%
Rolapitant	monkey NK1, Ki: 2.5 nM rat NK1, Ki: 78.6 nM rabbit NK1, Ki: 31.7 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM human NK1, Ki: 0.66 nM mouse NK1, Ki: 60.4 nM			98.65%
SB-222200			NK3	99.85%
Saredutant		NK2		98.02%
L-732138	NK1, IC₅₀: 2.3 nM			99.75%
Casopitant mesylate	NK1			99.84%
Osanetant			NK3	98.08%
Vofopitant dihydrochloride	NK1			99.11%
Orvepitant maleate	NK1, pKi: 10.2			99.99%
N-Acetyl-L-tryptophan	NK1			99.38%
Substance P TFA	NK1
Hemokinin 1, human	NK1	NK2	NK3	98.11%
Vapreotide	NK1			98.06%
L-733060 hydrochloride	NK1			≥99.0%
Biotin-Substance P	NK1			99.91%
Spantide I	NK1, Ki: 230 nM	NK2, Ki: 8150 nM		99.85%
Spantide II	NK1			98.01%
MEN 10207	NK1, pA2: 5.2	Tachykinin NK₂ Receptor, pA2: 7.9	NK3, pA2: 4.9	99.69%
Eprazinone dihydrochloride	NK1			≥98.0%
Eledoisin		NK2	NK3	99.05%
Fosnetupitant chloride monohydrochloride	hNK1, pKi: 9.5		hNK3, pKi: 6.1	99.70%
Vapreotide acetate	NK1			99.85%
[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)		NK2		99.83%
Rolapitant hydrochloride hydrate	monkey NK1, Ki: 2.5 nM rat NK1, Ki: 78.6 nM rabbit NK1, Ki: 31.7 nM gerbil NK1, Ki: 0.13 nM guinea pig NK1, Ki: 0.72 nM human NK1, Ki: 0.66 nM mouse NK1, Ki: 60.4 nM			98.25%
Nolpitantium	NK1
GR 159897		hNK2, pKi: 9.51 (CHO cell) NK2, pKi: 10 (Rat colon membrane)		≥99.0%
[MePhe7]-Neurokinin B			NK3, IC₅₀: 3 nM	98.87%
GR 87389		NK2
Hemokinin 1, human TFA	NK1	NK2	NK3
(D-Arg1,D-Pro2,D-Phe7,D-His9)-Substance P	NK1
GR 94800 TFA		NK2
[D-Trp2,7,9] Substance P	NK1, Ki: 1 μM	NK2, Ki: 1.3 μM	NK3, Ki: ~9 μM
[Pro9]-Substance P	NK1, EC₅₀: 0.93 nM
Scyliorhinin I	rat NK1, Ki: 0.9 nM	guinea pig NK-2, Ki: 2 nM
Rolapitant hydrochloride	monkey NK1, Ki: 2.5 rat NK1, Ki: 78.6 rabbit NK1, Ki: 31.7 gerbil NK1, Ki: 0.13 guinea pig NK1, Ki: 0.72 human NK1, Ki: 0.66 mouse NK1, Ki: 60.4
Acetylaszonalenin	NK1
Neurokinin Receptor (393-407), rat	NK1
γ-Neuropeptide (rabbit)		NK2
SSR 146977			NK3
L-741671	hNK1, Ki: 0.03 nM
L-760735	hNK1, IC₅₀: 0.19 nM			≥99.0%
SB 218795		hNK2, Ki: 1220 nM	hNK3, Ki: 13 nM	99.86%
(Trp7,β-Ala8)-Neurokinin A (4-10)			NK3
CP 122721 hydrochloride	human NK1, pIC₅₀: 9.8
SDZ NKT 343	hNK1, IC₅₀: 0.62 nM	hNK2, Ki: 0.52 μM	hNK3, Ki: 3.4 μM
Imnopitant	NK1
Phyllomedusin	NK1
CS-003 Free base	NK1, Ki: 2.3 nM	NK2, Ki: 0.54 nM
ZM 253270		Hamster Bladder NK-2, Ki: 2 nM
Befetupitant	NK1
Vestipitant	hNK1, pKi: 9.4
Physalaemin	NK1

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